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Enantiomer selective glucuronidation of the non-steroidal pure anti-androgen bicalutamide by human liver and kidney: role of the human UDP-glucuronosyltransferase (UGT)1A9 enzyme

Bicalutamide (Casodex®) is a non-steroidal pure anti-androgen used in the treatment of localized prostate cancer. It is a racemate drug and its activity resides in the (R)-enantiomer, with little in the (S)-enantiomer. A major metabolic pathway for bicalutamide is glucuronidation catalyzed by UDP-gl...

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מידע ביבליוגרפי
Main Authors: Grosse, Laurent, Campeau, Anne-Sophie, Caron, Sarah, Morin, Frédéric-Alexandre, Meunier, Kim, Trottier, Jocelyn, Caron, Patrick, Verreault, Mélanie, Barbier, Olivier
פורמט: Artigo
שפה:Inglês
יצא לאור: 2013
נושאים:
גישה מקוונת:https://ncbi.nlm.nih.gov/pmc/articles/PMC3815647/
https://ncbi.nlm.nih.gov/pubmed/23527766
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bcpt.12071
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