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A Medicinal Chemists’ Guide to Lead Optimization for Tuberculosis

Tuberculosis is a bacterial disease which predominantly affects the lungs and results in extensive tissue pathology. This pathology contributes to the complexity of drug development as it presents discrete microenvironments within which the bacterium resides, often under conditions where replication...

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Dettagli Bibliografici
Autori principali: Dartois, Véronique, Barry, Clifton E
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3789655/
https://ncbi.nlm.nih.gov/pubmed/23910985
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2013.07.006
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