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Design and synthesis of 3,5-disubstituted boron-containing 1,2,4-oxadiazoles as potential combretastatin A-4 (CA-4) analogs

We have designed and synthesized a small library of 3,5-disubstituted-1,2,4-oxadiazole containing combretastatin A-4 (CA-4) analogs. Our objective is to increase the efficacy of the CA-4 as an anti-tubulin and antimitotic agent by substituting the cis-alkene bond with one of its bioisosteres, the 1,...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Das, Bhaskar C., Tang, Xiang-Ying, Rogler, Patrick, Evans, Todd
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2012
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3771381/
https://ncbi.nlm.nih.gov/pubmed/24039307
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tetlet.2012.02.110
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