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ACK1 Tyrosine Kinase: Targeted Inhibition to Block Cancer Cell Proliferation

ACK1 tyrosine kinase, located on chromosome 3q29, is aberrantly activated, amplified or mutated in a wide variety of human cancers. While the deregulated kinase is oncogenic and its activation correlates with progression to metastatic stage, its inhibition causes cell cycle arrest, sensitizes cells...

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Autori principali: Mahajan, Kiran, Mahajan, Nupam P.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3750075/
https://ncbi.nlm.nih.gov/pubmed/23597703
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.canlet.2013.04.004
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