A carregar...

Ex-527 inhibits Sirtuins by exploiting their unique NAD(+)-dependent deacetylation mechanism

Sirtuins are protein deacetylases regulating metabolism and stress responses. The seven human Sirtuins (Sirt1–7) are attractive drug targets, but Sirtuin inhibition mechanisms are mostly unidentified. We report the molecular mechanism of Sirtuin inhibition by 6-chloro-2,3,4,9-tetrahydro-1H-carbazole...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Gertz, Melanie, Fischer, Frank, Nguyen, Giang Thi Tuyet, Lakshminarasimhan, Mahadevan, Schutkowski, Mike, Weyand, Michael, Steegborn, Clemens
Formato: Artigo
Idioma:Inglês
Publicado em: National Academy of Sciences 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3725051/
https://ncbi.nlm.nih.gov/pubmed/23840057
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1303628110
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!