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Ligand promiscuity through the eyes of the aminoglycoside N3 acetyltransferase IIa

Aminoglycoside-modifying enzymes (AGMEs) are expressed in many pathogenic bacteria and cause resistance to aminoglycoside (AG) antibiotics. Remarkably, the substrate promiscuity of AGMEs is quite variable. The molecular basis for such ligand promiscuity is largely unknown as there is not an obvious...

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Autors principals: Norris, Adrianne L, Serpersu, Engin H
Format: Artigo
Idioma:Inglês
Publicat: Blackwell Publishing Ltd 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3719086/
https://ncbi.nlm.nih.gov/pubmed/23640799
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/pro.2273
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