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Computational Exploration of Zinc Binding Groups for HDAC Inhibition

Histone deacetylases (HDACs) emerged as important drug targets in epigenetics. The most common HDAC inhibitors use hydroxamic acids as zinc binding groups despite unfavorable pharmacokinetic properties. A two-stage protocol of M05-2X calculations of a library of 48 fragments in a small model active...

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Bibliografiske detaljer
Main Authors: Chen, Kai, Xu, Liping, Wiest, Olaf
Format: Artigo
Sprog:Inglês
Udgivet: 2013
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3703144/
https://ncbi.nlm.nih.gov/pubmed/23586590
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jo400406g
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