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Predictions of In Vivo Prolactin Levels from In Vitro K(i) Values of D(2) Receptor Antagonists Using an Agonist–Antagonist Interaction Model

Prolactin elevation is a side effect of all currently available D(2) receptor antagonists used in the treatment of schizophrenia. Prolactin elevation is the result of a direct antagonistic D(2) effect blocking the tonic inhibition of prolactin release by dopamine. The aims of this work were to asses...

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Bibliographic Details
Main Authors: Petersson, Klas J., Vermeulen, An M., Friberg, Lena E.
Format: Artigo
Language:Inglês
Published: Springer US 2013
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC3675734/
https://ncbi.nlm.nih.gov/pubmed/23392818
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-012-9450-6
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