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Novel HSP90 inhibitor NVP-HSP990 targets cell cycle regulators to ablate Olig2-positive glioma tumor initiating cells

Genetic heterogeneity and signaling alterations diminish the effectiveness of single-agent therapies in glioblastoma multiforme (GBM). The heat shock protein HSP90 is a molecular chaperone for several signaling proteins that are deregulated in glioma cells. Thus, HSP90 inhibition may offer an approa...

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Autores principales: Fu, Jun, Koul, Dimpy, Yao, Jun, Wang, Shuzhen, Yuan, Ying, Colman, Howard, Sulman, Erik. P., Lang, Frederick. F., Yung, W.K. Alfred
Formato: Artigo
Lenguaje:Inglês
Publicado: 2013
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3655088/
https://ncbi.nlm.nih.gov/pubmed/23492364
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1158/0008-5472.CAN-12-2033
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