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Synthesis of Novel Analogs of Cabergoline: Improving Cardiovascular Safety by Removing 5-HT(2B) Receptor Agonism

[Image: see text] The dopamine agonist cabergoline has been used to treat prolactinomas, Parkinson’s disease, Cushing’s disease, and sexual dysfunction. However, its clinical use was severely curtailed when it was found that patients taking cabergoline had an increased risk of developing cardiac-val...

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Detalhes bibliográficos
Main Authors: Dosa, Peter I., Ward, Tim, Walters, Michael A., Kim, Suck Won
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2013
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3629922/
https://ncbi.nlm.nih.gov/pubmed/23606928
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml3003814
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