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Pharmacology and Structure of Isolated Conformations of the Adenosine A(2A) Receptor Define Ligand Efficacy

Using isolated receptor conformations crystal structures of the adenosine A(2A) receptor have been solved in active and inactive states. Studying the change in affinity of ligands at these conformations allowed qualitative prediction of compound efficacy in vitro in a system-independent manner. Agon...

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Detalhes bibliográficos
Main Authors: Bennett, Kirstie A., Tehan, Benjamin, Lebon, Guillaume, Tate, Christopher G., Weir, Malcolm, Marshall, Fiona H., Langmead, Christopher J.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2013
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3629831/
https://ncbi.nlm.nih.gov/pubmed/23429888
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.112.084509
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