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Synergistic Activation of p21-activated Kinase 1 by Phosphatidylinositol 4,5-Bisphosphate and Rho GTPases

Autoinhibited p21-activated kinase 1 (Pak1) can be activated in vitro by the plasma membrane-bound Rho GTPases Rac1 and Cdc42 as well as by the lipid phosphatidylinositol (4,5)-bisphosphate (PIP(2)). Activator binding is mediated by a GTPase-binding motif and an adjacent phosphoinositide-binding mot...

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Autors principals: Malecka, Kimberly A., Szentpetery, Zsofia, Peterson, Jeffrey R.
Format: Artigo
Idioma:Inglês
Publicat: American Society for Biochemistry and Molecular Biology 2013
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3610963/
https://ncbi.nlm.nih.gov/pubmed/23393142
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M112.428904
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