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Dissecting Fragment-Based Lead Discovery at the von Hippel-Lindau Protein:Hypoxia Inducible Factor 1α Protein-Protein Interface

Fragment screening is widely used to identify attractive starting points for drug design. However, its potential and limitations to assess the tractability of often challenging protein:protein interfaces have been underexplored. Here, we address this question by means of a systematic deconstruction...

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Main Authors: Molle, Inge Van, Thomann, Andreas, Buckley, Dennis L., So, Ernest C., Lang, Steffen, Crews, Craig M., Ciulli, Alessio
Format: Artigo
Jezik:Inglês
Izdano: 2012
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC3551621/
https://ncbi.nlm.nih.gov/pubmed/23102223
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2012.08.015
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