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Design and development of masked therapeutic antibodies to limit off-target effects: Application to anti-EGFR antibodies

Therapeutic antibodies frequently cause side effects by binding antigen in non-target tissues. Here we demonstrate a novel molecular design of antibodies that addresses this problem by reversibly “masking” antibody complementarity determining regions until they reach diseased tissues containing dise...

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Hlavní autoři: Donaldson, Joshua M., Kari, Csaba, Fragoso, Ruben C., Rodeck, Ulrich, Williams, John C.
Médium: Artigo
Jazyk:Inglês
Vydáno: 2009
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3546534/
https://ncbi.nlm.nih.gov/pubmed/19783899
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