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Creation of an HDAC-Based Yeast Screening Method for Evaluation of Marine-Derived Actinomycetes: Discovery of Streptosetin A()

A histone deacetylase (HDAC)-based yeast assay employing a URA3 reporter gene was applied as a primary screen to evaluate a marine-derived actinomycete extract library and identify human class III HDAC (SIRT) inhibitors. Based on the bioassay-guided purification, a new compound designated as strepto...

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Библиографические подробности
Главные авторы: Amagata, Taro, Xiao, Jing, Chen, Yi-Pei, Holsopple, Nicholas, Oliver, Allen G., Gokey, Trevor, Guliaev, Anton B., Minoura, Katsuhiko
Формат: Artigo
Язык:Inglês
Опубликовано: 2012
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC3532527/
https://ncbi.nlm.nih.gov/pubmed/23167691
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/np300640g
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