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Human NAD(P)H:quinone oxidoreductase type I (hNQO1) activation of quinone propionic acid trigger groups

NAD(P)H:quinone oxidoreductase type I (NQO1) is a target enzyme for triggered delivery of drugs at inflamed tissue and tumor sites, particularly those that challenge traditional therapies. Prodrugs, macromolecules, and molecular assemblies possessing trigger groups that can be cleaved by environment...

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Autors principals: Mendoza, Maria F., Hollabaugh, Nicole M., Hettiarachchi, Suraj U., McCarley, Robin L.
Format: Artigo
Idioma:Inglês
Publicat: 2012
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3525107/
https://ncbi.nlm.nih.gov/pubmed/22989153
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi300760u
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