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Human NAD(P)H:quinone oxidoreductase type I (hNQO1) activation of quinone propionic acid trigger groups

NAD(P)H:quinone oxidoreductase type I (NQO1) is a target enzyme for triggered delivery of drugs at inflamed tissue and tumor sites, particularly those that challenge traditional therapies. Prodrugs, macromolecules, and molecular assemblies possessing trigger groups that can be cleaved by environment...

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Autori principali: Mendoza, Maria F., Hollabaugh, Nicole M., Hettiarachchi, Suraj U., McCarley, Robin L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3525107/
https://ncbi.nlm.nih.gov/pubmed/22989153
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi300760u
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