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Jostling for Position: Optimizing Linker Location in the Design of Estrogen Receptor-targeting PROTACs

Estrogen receptor-alpha (ER) antagonists have been widely used for breast cancer therapy. Despite initial responsiveness, eventually hormone-sensitive ER-positive cancer cells develop resistance to ER antagonists. It has been shown that, in most of these resistant tumor cells, the ER is expressed an...

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Bibliografische gegevens
Hoofdauteurs: Cyrus, Kedra, Wehenkel, Marie, Choi, Eun-Young, Lee, Hyosung, Swanson, Hollie, Kim, Kyung-Bo
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2010
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Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3516907/
https://ncbi.nlm.nih.gov/pubmed/20512796
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201000146
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