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Comparison of the In Vivo Pharmacokinetics and In Vitro Dissolution of Raltegravir in HIV Patients Receiving the Drug by Swallowing or by Chewing

The pharmacokinetics of raltegravir (RAL) in HIV patients is characterized by high interpatient/intrapatient variability. We investigated the potential contribution of the drug pharmaceutical formulation to RAL pharmacokinetics. We first compared in vivo the pharmacokinetics of RAL for 67 patients t...

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Autors principals: Cattaneo, Dario, Baldelli, Sara, Cerea, Matteo, Landonio, Simona, Meraviglia, Paola, Simioni, Emanuela, Cozzi, Valeria, Fucile, Serena, Gazzaniga, Andrea, Clementi, Emilio, Galli, Massimo, Rizzardini, Giuliano, Gervasoni, Cristina
Format: Artigo
Idioma:Inglês
Publicat: American Society for Microbiology 2012
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3497176/
https://ncbi.nlm.nih.gov/pubmed/22964253
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.00942-12
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