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Direct Stereospecific Amination of Alkyl and Aryl Pinacol Boronates

The direct amination of alkyl and aryl pinacol boronates is accomplished with lithiated methoxyamine. This reaction directly provides aliphatic and aromatic amines, stereospecifically, and without preactivation of the boronate substrate.

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Detalles Bibliográficos
Autores principales: Mlynarski, Scott N., Karns, Alexander S., Morken, James P.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2012
Materias:
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3481838/
https://ncbi.nlm.nih.gov/pubmed/23002712
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja305448w
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