Загрузка...

Beta-endorphin: replacement of tyrosine in position 27 by tryptophan increases analgesic potency--preparation and properties of the 2-nitrophenylsulfenyl derivative.

An analog of human beta-endorphin with tryptophan in position 27 has been synthetized by the solid-phase method. Bioassay of the analog showed that it had almost 4 times the analgesic potency of the parent hormone but only 68% of the opiate receptor-binding activity. The peptide is the most potent a...

Полное описание

Сохранить в:
Библиографические подробности
Опубликовано в: :Proc Natl Acad Sci U S A
Главные авторы: Li, C H, Yamashiro, D, Nicolas, P
Формат: Artigo
Язык:Inglês
Опубликовано: National Academy of Sciences 1982
Предметы:
Online-ссылка:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC345895/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/6280164/
https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.79.4.1042
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!