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Inhibition of Na+/Ca2+ exchange in membrane vesicle and papillary muscle preparations from guinea pig heart by analogs of amiloride.

Na+/Ca2+ exchange is inhibited in both guinea pig cardiac membrane vesicles and papillary muscles in a concentration-dependent fashion by several analogs of the pyrazine diuretic amiloride. Structure/activity studies based on transport measurements in vesicles prepared from guinea pig left ventricle...

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Detalles Bibliográficos
Publicado en:Proc Natl Acad Sci U S A
Principais autores: Siegl, P K, Cragoe, E J, Trumble, M J, Kaczorowski, G J
Formato: Artigo
Idioma:Inglês
Publicado: National Academy of Sciences 1984
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Acceso en liña:https://ncbi.nlm.nih.govhttps://pmc.ncbi.nlm.nih.gov/articles/PMC345257/
https://ncbi.nlm.nih.govhttps://pubmed.ncbi.nlm.nih.gov/6587348/
https://ncbi.nlm.nih.govhttps://doi.org/10.1073/pnas.81.10.3238
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