Laddar...

Functionalized Congeners of 1,4-Dihydropyridines as Antagonist Molecular Probes for A(3) Adenosine Receptors

4-Phenylethynyl-6-phenyl-1,4-dihydropyridine derivatives are selective antagonists at human A(3) adenosine receptors, with K(i) values in a radioligand binding assay vs [(125)I]AB-MECA [N(6)-(4-amino-3-iodobenzyl)-5′-N-methylcarbamoyl-adenosine] in the submicromolar range. In this study, functionali...

Full beskrivning

Sparad:
Bibliografiska uppgifter
Huvudupphovsmän: Li, An-Hu, Chang, Louis, Ji, Xiao-duo, Melman, Neli, Jacobson, Kenneth A.
Materialtyp: Artigo
Språk:Inglês
Publicerad: 1999
Ämnen:
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC3446815/
https://ncbi.nlm.nih.gov/pubmed/10411465
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bc9900136
Taggar: Lägg till en tagg
Inga taggar, Lägg till första taggen!