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Covalent binding of a selective agonist irreversibly activates guinea pig coronary artery A(2) adenosine receptors

Experiments employing guinea pig heart Langendorff preparations compared the coronary vasoactivity of a functionalized congener of adenosine, 2-[(2-amino-ethylaminocarbonylethyl)phenylethylamino]-5′-N-ethylcarboxamidoadenosine, APEC, with the vasoactivity of the product of the reaction of APEC with...

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Autors principals: Niiya, Kazunori, Jacobson, Kenneth A., Silvia, Scott K., Olsson, Ray A.
Format: Artigo
Idioma:Inglês
Publicat: 1993
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3437322/
https://ncbi.nlm.nih.gov/pubmed/8321327
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