Conformationally Constrained Analogues of N'-(4-t-Butylbenzyl)-N-(4-Methylsulfonylaminobenzyl)Thiourea as TRPV1 Antagonists

A series of bicyclic analogues having indan and tetrahydronaphthalene templates in the A-region were designed as conformationally constrained analogues of our previously reported potent TRPV1 antagonists (1, 3). The activities for rat TRPV1 of the conformationally restricted analogues were moderatel...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Ryu, HyungChul, Lim, Ju-Ok, Kang, Dong Wook, Pearce, Larry V., Tran, Richard, Toth, Attila, Lee, Jeewoo, Blumberg, Peter M.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2008
Gaiak:
Article
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC3420357/
https://ncbi.nlm.nih.gov/pubmed/18406014
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2008.02.026
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