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Design, synthesis and in vitro antitumor activity evaluation of novel 4-pyrrylamino quinazoline derivatives

Here we describe the design and synthesis of two series of 4-pyrrylamino quinazolines as new analogues of the EGFR inhibitor Gefitinib. In vitro antitumor activity of these novel compounds against pancreatic (Miapaca2) and prostate (DU145) cancer cell lines was evaluated. Compared with the parental...

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Bibliografski detalji
Glavni autori: Wu, Xiaoqing, Li, Mingdong, Tang, Wenhua, Zheng, Youguang, Lian, Jiqin, Xu, Liang, Ji, Min
Format: Artigo
Jezik:Inglês
Izdano: 2011
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC3412131/
https://ncbi.nlm.nih.gov/pubmed/21895983
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/j.1747-0285.2011.01234.x
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