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First-pass metabolism via UDP-glucuronosyltransferase: a barrier to oral bioavailability of phenolics
Glucuronidation mediated by UDP-glucuronosyltransferases (UGTs) is a significant metabolic pathway that facilitates efficient elimination of numerous endo- and xenobiotics including phenolics. UGT genetic deficiency and polymorphisms or inhibition of glucuronidation by concomitant use of drugs are a...
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| Главные авторы: | , , , , |
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| Формат: | Artigo |
| Язык: | Inglês |
| Опубликовано: |
2011
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| Предметы: | |
| Online-ссылка: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3409645/ https://ncbi.nlm.nih.gov/pubmed/21484808 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jps.22568 |
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