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Regulation of drug resistance by human pregnane X receptor in breast cancer

Drug resistance is a significant barrier to an effective treatment of breast cancer. Human pregnane X receptor (hPXR), an orphan nuclear receptor known for its activation by many important clinical drugs, is a major transcription factor of drug metabolism enzymes (DMEs), such as cytochrome P450 3A4...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Chen, Yakun, Tang, Yong, Chen, Shuqing, Nie, Daotai
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2009
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3392171/
https://ncbi.nlm.nih.gov/pubmed/19746521
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