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Synthesis and evaluation of indole-based chalcones as inducers of methuosis, a novel type of non-apoptotic cell death

Methuosis is a novel caspase-independent form of cell death in which massive accumulation of vacuoles derived from macropinosomes ultimately causes cells to detach from the substratum and rupture. We recently described a chalcone-like compound, 3-(2-methyl-1H indol-3-yl)-1-(4-pyridinyl)-2-propen-1-o...

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Autori principali: Robinson, Michael W., Overmeyer, Jean H., Young, Ashley M., Erhardt, Paul W., Maltese, William A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2012
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3314534/
https://ncbi.nlm.nih.gov/pubmed/22335538
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm201006x
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