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Development of Potent and Selective Inhibitors of Aldo-Keto Reductase 1C3 (type 5 17β-Hydroxysteroid Dehydrogenase) Based on N-Phenyl-Aminobenzoates and Their Structure Activity Relationships

Aldo-keto reductase 1C3 (AKR1C3; type 5 17β-hydroxysteroid dehydrogenase) is overexpressed in castrate resistant prostate cancer (CRPC) and is implicated in the intratumoral biosynthesis of testosterone and 5α-dihydrotestosterone. Selective AKR1C3 inhibitors are required since compounds should not i...

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Detalhes bibliográficos
Main Authors: Adeniji, Adegoke O., Twenter, Barry M., Byrns, Michael C., Jin, Yi, Chen, Mo, Winkler, Jeffrey D., Penning, Trevor M.
Formato: Artigo
Idioma:Inglês
Publicado em: 2012
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3298089/
https://ncbi.nlm.nih.gov/pubmed/22263837
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm201547v
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