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Virtual Screening Targeting the Urokinase Receptor, Biochemical and Cell-Based Studies, Synthesis, Pharmacokinetic Characterization, and Effect on Breast Tumor Metastasis

Virtual screening targeting the urokinase receptor (uPAR) led to (3R)-4-cyclohexyl-3-(hexahydrobenzo[d][1,3]dioxol-5-yl)-N-((hexahydrobenzo[d][1,3]dioxol-5-yl)methyl)butan-1-aminium 1 (IPR-1) and 4-(4-((3,5-dimethylcyclohexyl)carbamoyl)-2-(4-isopropylcyclohexyl)pyrazolidin-3-yl)piperidin-1-ium 3 (IP...

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Detalhes bibliográficos
Main Authors: Wang, Fang, Li, Jing, Sinn, Anthony L., Knabe, William Eric, Khanna, May, Jo, Inha, Silver, Jayne M., Oh, Kyungsoo, Li, Liwei, Sandusky, George E., Sledge, George W., Nakshatri, Harikrishna, Jones, David R., Pollok, Karen E., Meroueh, Samy O.
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3280887/
https://ncbi.nlm.nih.gov/pubmed/21851064
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm200782y
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