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Study of the role of “gatekeeper” mutations V654A and T670I of c-kit kinase in the interaction with inhibitors by means mixed molecular dynamics/docking approach

The over-expression of c-kit proto-oncogene has been reported in hematopoietic cells, small cell lung cancer, and gastrointestinal stromal tumors. The clinical importance of c-kit expression in tumors focused the research towards inhibitors of this tyrosine kinase. Imatinib (Gleevec®) was the first...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: Tutone, Marco, Lauria, Antonino, Almerico, Anna Maria
Format: Artigo
Sprache:Inglês
Veröffentlicht: Biomedical Informatics 2011
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3280498/
https://ncbi.nlm.nih.gov/pubmed/22355224
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