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An Orally Bioavailable c-Met Kinase Inhibitor Potently Inhibits Brain Tumor Malignancy and Growth

The receptor tyrosine kinase, c-Met and its ligand hepatocyte growth factor (HGF) are important regulators of malignancy in human cancer including brain tumors. c-Met is frequently activated in brain tumors and has emerged as a promising target for molecular therapies. Recently, an orally bioavailab...

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Detalhes bibliográficos
Main Authors: Guessous, Fadila, Zhang, Ying, diPierro, Charles, Marcinkiewicz, Lukasz, Sarkaria, Jann, Schiff, David, Buchanan, Sean, Abounader, Roger
Formato: Artigo
Idioma:Inglês
Publicado em: 2010
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3278215/
https://ncbi.nlm.nih.gov/pubmed/20015006
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