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Oleanane triterpenoid CDDO-Me inhibits Akt activity without affecting PDK1 kinase or PP2A phosphatase activity in cancer cells

Our previous studies have shown that methyl-2-cyano-3,12-dioxooleana-1,9(11)-dien-28-oate (CDDO-Me), a oleanane synthetic triterpenoid induces apoptosis in prostate cancer cells by inhibiting the Akt/NF-κB/mTOR signaling cascade; however, the mechanism by which CDDO-Me inhibits Akt/NF-κB/mTOR signal...

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Autors principals: Liu, Yongbo, Gao, Xiaohua, Deeb, Dorrah, Gautam, Subhash C.
Format: Artigo
Idioma:Inglês
Publicat: 2011
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3264055/
https://ncbi.nlm.nih.gov/pubmed/22177954
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bbrc.2011.12.007
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