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A short update on the structure of drug binding sites on neurotransmitter transporters

BACKGROUND: The dopamine (DAT), noradrenalin (NET) and serotonin (SERT) transporters are molecular targets for different classes of psychotropic drugs. Cocaine and the SSRI (S)-citalopram block neurotransmitter reuptake competitively, but while cocaine is a non-selective reuptake inhibitor, (S)-cita...

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Autors principals: Gabrielsen, Mari, Sylte, Ingebrigt, Dahl, Svein G, Ravna, Aina W
Format: Artigo
Idioma:Inglês
Publicat: BioMed Central 2011
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3259071/
https://ncbi.nlm.nih.gov/pubmed/22192271
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1186/1756-0500-4-559
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