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Palmitoylation influences the function and pharmacology of sodium channels

Palmitoylation is a common lipid modification known to regulate the functional properties of various proteins and is a vital step in the biosynthesis of voltage-activated sodium (Nav) channels. We discovered a mutation in an intracellular loop of rNav1.2a (G1079C), which results in a higher apparent...

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Autori principali: Bosmans, Frank, Milescu, Mirela, Swartz, Kenton J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: National Academy of Sciences 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3250191/
https://ncbi.nlm.nih.gov/pubmed/22123950
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1108497108
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