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A novel compound inhibits rHDL assembly and blocks nascent HDL biogenesis downstream of apoAI binding to ABCA1 expressing cells

OBJECTIVE: Nascent high-density lipoprotein (HDL) particles form from cellular lipids and extracellular lipid-free apolipoprotein AI (apoAI) in a process mediated by ATP-binding cassette transporter A1 (ABCA1). We have sought out compounds that inhibit nascent HDL biogenesis without affecting ABCA1...

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Autori principali: Lyssenko, Nicholas N., Brubaker, Gregory, Smith, Bradley D., Smith, Jonathan D.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3197940/
https://ncbi.nlm.nih.gov/pubmed/21836073
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1161/ATVBAHA.111.234906
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