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Intestinal Absorption of Novel-Dipeptide Prodrugs of Saquinavir in Rats

Saquinavir (SQV) was the first human immuno-virus-1 (HIV-1) protease inhibitor approved by FDA. However, P-glycoprotein (P-gp), an efflux pump limits its oral and brain bioavailabilities. The objective of this study is to investigate whether prodrug modification of SQV to dipeptide prodrugs Valine-V...

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Bibliografske podrobnosti
Main Authors: Jain, Ritesh, Duvvuri, Sridhar, Kansara, Viral, Mandava, Nanda Kishore, Mitra, Ashim K.
Format: Artigo
Jezik:Inglês
Izdano: 2006
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC3166959/
https://ncbi.nlm.nih.gov/pubmed/17207946
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ijpharm.2006.11.058
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