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Synthesis and PET studies of [(11)C-cyano]letrozole (Femara(®)), an aromatase inhibitor drug

INTRODUCTION: Aromatase, a member of the cytochrome P450 family, converts androgens such as androstenedione and testosterone to estrone and estradiol respectively. Letrozole (1-[bis-(4-cyanophenyl)methyl]-1H-1,2,4-triazole, Femara(®)) is a high affinity aromatase inhibitor (K(i)=11.5 nM) which has F...

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Bibliographische Detailangaben
Hauptverfasser: Kil, Kun-Eek, Biegon, Anat, Ding, Yu-Shin, Fischer, Andre, Ferrieri, Richard A., Kim, Sung Won, Pareto, Deborah, Schueller, Michael J., Fowler, Joanna S.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2009
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC3161428/
https://ncbi.nlm.nih.gov/pubmed/19217534
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.nucmedbio.2008.11.010
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