Nalaganje...

Design and Synthesis of 3,5-Disubstituted 1,2,4-Oxadiazole Containing Retinoids from a Retinoic Acid Receptor Agonist

We previously synthesized novel retinoid libraries, and after screening for bioactivity found one compound BT10 that functions as a specific agonist for retinoic acid receptors. This lead compound was further derivatized using SAR and LRD to obtain 3,5-disubstituted-1,2,4-oxadiazole-containing retin...

Popoln opis

Shranjeno v:
Bibliografske podrobnosti
Main Authors: Das, Bhaskar C., Tang, Xiang-Ying, Sanyal, Swarnava, Mohapatra, Seetaram, Rogler, Patrick, Nayak, Sabita, Evans, Todd
Format: Artigo
Jezik:Inglês
Izdano: 2011
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC3135900/
https://ncbi.nlm.nih.gov/pubmed/21765558
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tetlet.2011.03.011
Oznake: Označite
Brez oznak, prvi označite!