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Identifying selective inhibitors against human cytosolic sialidase NEU2 by substrate specificity studies

Aberrant expression of human sialidases has been shown to associate with various pathological conditions. Despite the effort in sialidase inhibitor design, less attention has been paid to designing specific inhibitors against human sialidases and characterizing the substrate specificity of different...

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Detalhes bibliográficos
Main Authors: Li, Yanhong, Cao, Hongzhi, Yu, Hai, Chen, Yi, Lau, Kam, Qu, Jingyao, Thon, Vireak, Sugiarto, Go, Chen, Xi
Formato: Artigo
Idioma:Inglês
Publicado em: 2011
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC3114945/
https://ncbi.nlm.nih.gov/pubmed/21206954
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c0mb00244e
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