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Trypanocidal Furamidine Analogues: Influence of Pyridine Nitrogens on Trypanocidal Activity, Transport Kinetics, and Resistance Patterns

Current therapies for human African trypanosomiasis (HAT) are unsatisfactory and under threat from emerging drug resistance linked to the loss of transporters, e.g., the P2 aminopurine transporter (TbAT1). Here we compare the uptake and trypanocidal properties of furamidine (DB75), recently evaluate...

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Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Ward, Christopher P., Wong, Pui Ee, Burchmore, Richard J., de Koning, Harry P., Barrett, Michael P.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: American Society for Microbiology 2011
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC3088251/
https://ncbi.nlm.nih.gov/pubmed/21402852
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01551-10
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