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(18)F-Labeled GRPR Agonists and Antagonists: A Comparative Study in Prostate Cancer Imaging

Radiolabeled bombesin analogs are promising probes for cancer imaging of gastrin-releasing peptide receptor (GRPR). In this study, we developed (18)F-labeled GRPR agonists and antagonists for positron emission tomography (PET) imaging of prostate cancer. GRPR antagonists ATBBN (D-Phe-Gln-Trp-Ala-Val...

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Autori principali: Yang, Min, Gao, Haokao, Zhou, Yaru, Ma, Ying, Quan, Qimeng, Lang, Lixin, Chen, Kai, Niu, Gang, Yan, Yongjun, Chen, Xiaoyuan
Natura: Artigo
Lingua:Inglês
Pubblicazione: Ivyspring International Publisher 2011
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3086613/
https://ncbi.nlm.nih.gov/pubmed/21544226
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