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Integration of Preclinical and Clinical Data with Pharmacokinetic Modeling and Simulation to Evaluate Fexofenadine as a Probe for Hepatobiliary Transport Function

PURPOSE: The suitability of fexofenadine as a probe substrate to assess hepatobiliary transport function in humans was evaluated by pharmacokinetic modeling/simulation and in vitro/in situ studies using chemical modulators. METHODS: Simulations based on a pharmacokinetic model developed to describe...

Täydet tiedot

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Bibliografiset tiedot
Päätekijät: Swift, Brandon, Tian, Xianbin, Brouwer, Kim L. R.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2009
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC3083979/
https://ncbi.nlm.nih.gov/pubmed/19495943
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11095-009-9909-z
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