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An efficient methodology to substituted furans via oxidation of functionalized α-diazo-β-ketoacetates

DMDO oxidation of functionalized α-diazo-β-ketoacetates, formed by zinc triflate catalyzed Mukaiyama-aldol condensation of methyl diazoacetoacetate with aldehydes, occurred in quantitative yield to form dihydrofuranols that undergo acid catalyzed dehydration under mild conditions to generate 3-metho...

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Main Authors: Truong, Phong, Xu, Xinfang, Doyle, Michael P.
Formato: Artigo
Idioma:Inglês
Publicado: 2011
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC3080702/
https://ncbi.nlm.nih.gov/pubmed/21516185
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tetlet.2010.11.166
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