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Ligand selectivity by seeking hydrophobicity in thyroid hormone receptor

Selective therapeutics for nuclear receptors would revolutionize treatment for endocrine disease. Specific control of nuclear receptor activity is challenging because the internal cavities that bind hormones can be virtually identical. Only one highly selective hormone analog is known for the thyroi...

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Autori principali: Borngraeber, Sabine, Budny, Mary-Jane, Chiellini, Grazia, Cunha-Lima, Suzana T., Togashi, Marie, Webb, Paul, Baxter, John D., Scanlan, Thomas S., Fletterick, Robert J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: National Academy of Sciences 2003
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC307572/
https://ncbi.nlm.nih.gov/pubmed/14673100
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.2136689100
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