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Inhibition of amyloidogenesis by non-steroidal anti-inflammatory drugs and their hybrid nitrates

Poor blood-brain barrier penetration of non-steroidal anti-inflammatory drugs (NSAIDs) has been blamed for the failure of the selective amyloid lowering agent (SALA) R-flurbiprofen in phase 3 clinical trials for Alzheimer’s disease (AD). NO-donor NSAIDs (NO-NSAIDs) provide an alternative, gastric-sp...

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Autores principales: Schiefer, Isaac T., Abdul-Hay, Samer, Wang, Huali, Vanni, Michael, Qin, Zhihui, Thatcher, Gregory R. J.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2011
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC3072465/
https://ncbi.nlm.nih.gov/pubmed/21405086
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm101450p
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