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Reduced fidelity of branch point recognition and alternative splicing induced by the anti-tumor drug spliceostatin A

Spliceostatin A (SSA) is a stabilized derivative of a Pseudomonas bacterial fermentation product that displays potent anti-proliferative and anti-tumor activities in cancer cells and animal models. The drug inhibits pre-mRNA splicing in vitro and in vivo and binds SF3b, a protein subcomplex of U2 sm...

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Autors principals: Corrionero, Anna, Miñana, Belén, Valcárcel, Juan
Format: Artigo
Idioma:Inglês
Publicat: Cold Spring Harbor Laboratory Press 2011
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3049286/
https://ncbi.nlm.nih.gov/pubmed/21363963
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1101/gad.2014311
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