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Structural determinants of ligand imprinting: A molecular dynamics simulation study of subtilisin in aqueous and apolar solvents

The phenomenon known as “ligand imprinting” or “ligand-induced enzyme memory” was first reported in 1988, when Russell and Klibanov observed that lyophilizing subtilisin in the presence of competitive inhibitors (that were subsequently removed) could significantly enhance its activity in an apolar s...

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Autors principals: Lousa, Diana, Baptista, António M, Soares, Cláudio M
Format: Artigo
Idioma:Inglês
Publicat: Wiley Subscription Services, Inc., A Wiley Company 2011
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC3048422/
https://ncbi.nlm.nih.gov/pubmed/21280129
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/pro.569
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