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A Novel PET Marker for In Vivo Quantification of Myelination
C-11-Labeled N-methyl-4,4′-diaminostilbene ([(11)C]MeDAS) was synthesized and evaluated as a novel radiotracer for in vivo microPET imaging of myelination. [(11)C]MeDAS exhibits optimal lipophilicity for brain uptake with a logPoct value of 2.25. Both in vitro and ex vivo staining exhibited MeDAS ac...
Αποθηκεύτηκε σε:
| Κύριοι συγγραφείς: | , , , , , , , , , , |
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| Μορφή: | Artigo |
| Γλώσσα: | Inglês |
| Έκδοση: |
2010
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| Θέματα: | |
| Διαθέσιμο Online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC3044472/ https://ncbi.nlm.nih.gov/pubmed/21071233 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2010.10.018 |
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